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R. Abed Ali Abdine; G. Hedouin, F. Colobert; J. Wencel-Delord

Metal-Catalyzed Asymmetric Hydrogenation of C═N Bonds Journal Article

ACS Catalysis 2021, 11, 215-247.

Links | Tags: SYNCAT


G. Hedouin; Q. Dherbassy; J. Wencel-Delord; F. colobert

An Improvement of the Synthesis of (1R,2S,5R)-(–)-Menthyl (S)-p-Toluenesulfinate Journal Article

SynOpen 2021, 05, 65-67.

Links | Tags: SYNCAT



J. Frey; S. Choppin; F. Colobert; J. Wencel-Delord

Towards Atropoenantiopure N–C Axially Chiral Compounds via Stereoselective C– N Bond Formation Journal Article

Chimia 2020, 74, 883-889.

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J. Wencel-Delord; F. Colobert

Challenging Atroposelective C–H Arylation Journal Article

SynOpen 2020, 04, 107-115.

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T. Guérin; N. V. Pikun; R. Morioka; A. Panossian; G. Hanquet; F. R. Leroux

Synthesis and use of trifluoromethylthiolated ketenimines Journal Article

Chemistry a European Journal 2020, 26, 14852-14855.

Links | Tags: COHA, SYNCAT


J. Wencel-Delord

Decorating and diversifying drugs Journal Article

Nature Chemistry 2020, 12, 505-506.

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R. Mei; U. Dhawa; R.C. Samanta; W. Ma; J. Wencel-Delord; L. Ackermann

Cobalt-Catalyzed Oxidative C−H Activation: Strategies and Concepts Journal Article

ChemSusChem 2020, 13, 3306-3356.

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J. Frey; A. Malekafzali; I. Delso; S. Choppin; F. Colobert; J. Wencel-Delord

Enantioselective Synthesis of N-C Axially Chiral Compounds by Cu-catalyzed Atroposelective Aryl Amination Journal Article

Angewandte Chemie International Edition 2020, 59, 8844-8848.

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N. Jacob; L. Guillemard; J. Wencel-Delord

Highly Efficient Synthesis of Hindered 3-Azoindoles via Metal-Free C–H Functionalization of Indoles Journal Article

Synthesis 2020, 52, 574–580.

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M. Hlaváč; L. Kováčiková; M. Šoltésová Prnová; P. Šramel; G. Addová; M. Májeková; G. Hanquet; A. Boháč; M. Štefek

Development of Novel Oxotriazinoindole Inhibitors of Aldose Reductase: Isosteric Sulfur/Oxygen Replacement in the Thioxotriazinoindole Cemtirestat Markedly Improved Inhibition Selectivity Journal Article

Journal of Medicinal Chemistry 2020, 63, 369-381.

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P. Massé; S. Choppin; L. Chiummiento; G. Hanquet; F. Colobert

Unintended Formation of a 26-Membered Cycle in the Course of a Novel Approach to Myricanol, a Strained [7,0]-Metacyclophane Journal Article

Synlett 2020, 31, 559-564.

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Y. Qiu; S. Chan; L. Lin; T. Lam Shek; T. Fung Tsang; Y. Zhang; M. Ip; P. Kay-sheung Chan; N. Blanchard; G. Hanquet; Z. Zuo; X. Yang; C. Ma

Nusbiarylins, a new class of antimicrobial agents: Rational design of bacterial transcription inhibitors targeting the interaction between the NusB and NusE proteins Journal Article

Bioorganic Chemistry 2019, 92, 103203.

Links | Tags: BSM, SYNCAT


T. Anitha; K. Chinna Ashalu; M. Sandeep; A. Mohd; J. Wencel‐Delord; F. Colobert; K. Rajender Reddy

LiI/TBHP Mediated Oxidative Cross‐Coupling of P(O)–H Compounds with Phenols and Various Nucleophiles: Direct Access to the Synthesis of Organophosphates Journal Article

European Journal of Organic Chemistry 2019, 2019, 7463-7474.

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F. Colobert; J. Wencel-Delord

C-H Activation for Asymmetric Synthesis Book

Wiley-VCH, 2019, ISBN: 978-3-527-34340-9.

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J. Loup; U. Dhawa; F. Pesciaioli; J. Wencel‐Delord; L. Ackermann

Enantioselective C−H Activation with Earth‐Abundant 3d Transition Metals Journal Article

Angewandte Chemie International Edition 2019, 58, 12803-12818.

Abstract | Links | Tags: SYNCAT


Y. Qiu; S. Ting Chan; L. Lin; T. L. Shek; T. F. Tsang; N. Barua; Y. Zhang; M. Ip; P. K.-S. Chan; N. Blanchard; G. Hanquet; Z. Zuo; X. Yang; C. Ma

Design, synthesis and biological evaluation of antimicrobial diarylimine and –amine compounds targeting the interaction between the bacterial NusB and NusE proteins Journal Article

European Journal of Medicinal Chemistry 2019, 178, 214 - 231.

Abstract | Links | Tags: BSM, SYNCAT


S Jerhaoui; J-P Djukic; J Wencel-Delord; F Colobert

Asymmetric, Nearly Barrierless C(sp3)–H Activation Promoted by Easily-Accessible N-Protected Aminosulfoxides as New Chiral Ligands Journal Article

ACS Catalysis 2019, 9, 2532-2542.

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A Srinivasulu; B Shantharjun; D Vani; Chinna K Ashalu; A Mohd; J Wencel-Delord; F Colobert; R K Reddy

Iron-Catalyzed Minisci Type Acetylation of N-Heteroarenes Mediated by CH(OEt)3/TBHP Journal Article

European Journal of Organic Chemistry 2019, 2019, 1815-1819.

Abstract | Links | Tags: SYNCAT



F. Ulm; A.I. Poblador-Bahamonde; S. Choppin; S. Bellemin-Laponnaz M.J. Chetcuti; T. Achard; V. Ritleng

Synthesis, characterization, and catalytic application in aldehyde hydrosilylation of half-sandwich nickel complexes bearing (κ1-C)- and hemilabile (κ2-C,S)-thioether-functionalised NHC ligands Journal Article

Dalton Transactions 2018, 47, 17134-17145 .

Links | Tags: COA, SYNCAT


L. Guillemard; F. Colobert; J. Wencel-Delord

Visible-Light-Triggered, Metal- and Photocatalyst-Free Acylation of N-Heterocycles Journal Article

Advanced Synthesis & Catalysis 2018, 360, 4184-4190.

Abstract | Links | Tags: SYNCAT


A. Bochicchio; L. Schiavo; L. Chiummiento; P. Lupattelli; M. Funicello; G. Hanquet; S. Choppin; F. Colobert

Convergent total synthesis of (±) myricanol, a cyclic natural diarylheptanoid Journal Article

Organic & Biomolecular Chemistry 2018, 16, 8859-8869 .

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Q. Dherbassy; J. Wencel-Delord; F. Colobert

Atroposelective arylation of biaryls by C-H activation Journal Article

Tetrahedron 2018, 74, 6205 - 6212.

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C. Batisse; A. Panossian; G. Hanquet; and F. R. Leroux

Access towards enantiopure α,α-difluoromethyl alcohols by means of sulfoxides as traceless chiral auxiliaries Journal Article

Chemical Communications 2018, 54, 10423-10426 .

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C. Sambiagio; D. Schönbauer; R. Blieck; T. Dao-Huy; G. Pototschnig; P. Schaaf; T. Wiesinger; M. Farooq Zia; J. Wencel-Delord; T. Besset; B. U. W. Maesa; Michael Schnürch

A comprehensive overview of directing groups applied in metal-catalysed C–H functionalisation chemistry Journal Article

Chemical Society Reviews 2018, 47, 6603-6743.

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L. Schiavo; L. Lebedel; P. Massé; S. Choppin; G. Hanquet

Access to Wieland–Miescher Diketone-Derived Building Blocks by Stereoselective Construction of the C-9 Quaternary Carbon Center Using the Mukaiyama Aldol Reaction Journal Article

The Journal of Organic Chemistry 2018, 83, 6247-6258.

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D. Meidlinger; L. Marx; C. Bordeianu; S. Choppin; F. Colobert; A. Speicher

Access to the Enantiopure Axially Chiral Cyclophane Isoplagiochin D through Atropo-diastereoselective Heck Coupling Journal Article

Angewandte Chemie International Edition 2018, 57, 9160-9164.

Abstract | Links | Tags: SYNCAT


Q. Dherbassy; J.-P. Djukic; J. Wencel‐Delord; F. Colobert

Two Stereoinduction Events in One C−H Activation Step: A Route towards Terphenyl Ligands with Two Atropisomeric Axes Journal Article

Angewandte Chemie 2018, 130, 4758-4762.

Abstract | Links | Tags: SYNCAT


C. Selvam; I. A Lemasson; I. Brabet; N. Oueslati; B. Karaman; A. Cabaye; A. S Tora; B. Commare; T. Courtiol; S. Cesarini; I. McCort-Tranchepain; D. Rigault; L. Mony; T. Bessiron; H. McLean; F. R Leroux; F. Colobert; H. Daniel; A. Goupil-Lamy; H.-O. Bertrand; C. Goudet; J.-P. Pin; F. C Acher

Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites Journal Article

Journal of Medicinal Chemistry 2018, 61, 1969-1989.

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H. Norouzi-Arasi; X. J. Salom-Roig; S.Lanners; G. Hanquet

First Total Synthesis of Pamamycin-621D Journal Article

Current Organic Synthesis 2018, 15, 105-109.

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James Rae; Johanna Frey; Soufyan Jerhaoui; Sabine Choppin; Joanna Wencel-Delord; Françoise Colobert

Synthesis of Axially Chiral C–N Scaffolds via Asymmetric Coupling with Enantiopure Sulfinyl Iodanes Journal Article

ACS Catalysis 2018, 8, 2805-2809.

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S. Jerhaoui; P. Poutrel; J.-P. Djukic; J. Wencel-Delord; F. Colobert

Stereospecific C-H activation as a key step for the asymmetric synthesis of various biologically active cyclopropanes Journal Article

Organic Chemistry Frontiers 2018, 5, 409-414.

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J. Wencel-Delord; F. Colobert

Super-reactive catalyst for bond cleavage Journal Article

Nature 2017, 551, 447-448.

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G. Della Sala; M. Sicignano; R. Schettini; F. De Riccardis; L. Cavallo; Y. Minenkov; C. Batisse; G. Hanquet; F. R. Leroux; I. Izzo

Switchable Diastereoselectivity in the Fluoride-Promoted Vinylogous Mukaiyama–Michael Reaction of 2-[(Trimethylsilyl)oxy]furan Catalyzed by Crown Ethers Journal Article

Journal of Organic Chemistry 2017, 82, 6629–6637.

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M. Murár; J. Dobiaš; P. Šramel; G. Addová; G. Hanquet; A. Boháč

Novel CLK1 inhibitors based on N-aryloxazol-2-amine skeleton - A possible way to dual VEGFR2 TK/CLK ligands Journal Article

European Journal of Medicinal Chemistry 2017, 126, 754 - 761.

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L. Schiavo; L. Jeanmart; S. Lanners; S. Choppin; G. Hanquet

FeCl3.6H2O/acetaldehyde, a versatile system for the deprotection of ketals and acetals via a transacetalization process Journal Article

New Journal of Chemistry 2017, 41, 1421-1424.

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D. C. Kahraman; G. Hanquet; L. Jeanmart; S. Lanners; P. Sramel; A. Bohac; R. Cetin-Atalay

Quinoides and VEGFR2 TKIs influence the fate of hepatocellular carcinoma and its cancer stem cells Journal Article

MedChemComm 2017, 8, 81-87.

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P. B. Arockiam; L. Guillemard; J. Wencel-Delord

Regiodivergent Visible Light-Induced C–H Functionalization of Quinolines at C-5 and C-8 under Metal-, Photosensitizer- and Oxidant-Free Conditions Journal Article

Advanced Synthesis & Catalysis 2017, 359, 2571-2579.

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S. Jerhaoui; J.-P. Djukic; J. Wencel-Delord; F. Colobert

Stereoselective Sulfinyl Aniline-Promoted Pd-Catalyzed C−H Arylation and Acetoxylation of Aliphatic Amides Journal Article

Chemistry – A European Journal 2017, 23, 15594-15600.

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E. Evain-Bana; L. Schiavo; C. Bour; D. A. Lanfranchi; S. Berardozzi; F. Ghirga; D. Bagrel; B. Botta; G. Hanquet; M. Mori

Synthesis, biological evaluation and molecular modeling studies on novel quinonoid inhibitors of CDC25 phosphatases Journal Article

Journal of Enzyme Inhibition and Medicinal Chemistry 2017, 32, 113-118.

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